JAMA Internal Medicine · March 2026

Extended-Release vs Sublingual Buprenorphine in Pregnancy

A Randomized Clinical Trial Through 12 Months Post Partum

N = 140
Participants
13 Sites
US Centers
2020–2024
Enrollment Period
NCT03918850
ClinicalTrials.gov

Winhusen TJ et al. JAMA Intern Med. doi:10.1001/jamainternmed.2026.0057

Background

Why Consider Extended-Release Buprenorphine?

Challenge 1
💊

Diversion & Misuse

Daily sublingual tablets carry risk of diversion and non-prescribed use.

Challenge 2
📉

Adherence Barriers

Daily dosing during pregnancy is associated with poor adherence rates.

Challenge 3
🔄

Peak-Trough Effects

Plasma levels fall during pregnancy, inadequately suppressing cravings.

Extended-release buprenorphine (Brixadi/CAM2038) provides stable plasma levels via weekly subcutaneous injection — potentially addressing all three challenges.

Methods

Trial Design

1
Enrollment
Adults with OUD, singleton pregnancy 6–30 wks GA
2
Randomization
1:1 allocation · Balanced on site & GA
3
Pregnancy Phase
Weekly ER-BUP injection vs daily SL-BUP
4
Delivery
Infant NOWS monitoring & outcomes
5
Post Partum
12-month follow-up · Monthly visits
Extended-Release (n=69)

Brixadi 24 mg/wk SC injection during pregnancy; monthly option post partum if not breastfeeding

Sublingual (n=71)

Generic buprenorphine tablets or buprenorphine/naloxone film; target 16 mg/day

Open-label, noninferiority RCT · 13 US outpatient peripartum OUD treatment sites · July 2020 – October 2024

Study Population

Participant Characteristics

Mean Age
31.2 yrs
SD 4.6 · Range 18–41
Mean GA at Enrollment
21.1 wks
SD 6.5
Already on Buprenorphine
98.6%
Clinically stable population
OUD (DSM-5, past 12 mo)
75.7%
Moderate or severe
Polysubstance Use
85%
Cotinine positive; 14% amphetamine
Study Completion
81%
Through 12 months post partum

82.9% White · 7.1% Black · 7.1% Hispanic · 10% Additional groups

Primary Outcome · Pregnancy

Illicit Opioid Abstinence During Pregnancy

Extended-Release
82.5%
Negative urine samples
Superior · P = .009
vs
Sublingual
72.6%
Negative urine samples

Noninferiority was demonstrated; superiority testing confirmed ER-BUP advantage.
Buprenorphine adherence was high and similar in both groups (~85%).

Primary outcome: proportion of weekly UDS negative for fentanyl, morphine, heroin, oxycodone, and other illicit opioids. Missing samples imputed as positive.

Key Secondary Outcome · Post Partum

Illicit Opioid Abstinence Post Partum

Extended-Release
60.2%
Negative urine samples
No Difference · P = .45
vs
Sublingual
59.5%
Negative urine samples
Postpartum Adherence
ER-BUP: 69.3% · SL-BUP: 75.5%
Difference not significant (P = .30)
Medication Discontinuation
35% postpartum vs 10% during pregnancy
Custody demands & CPS involvement cited

90% of participants retained maternal custody · 36% had open CPS cases

Infant Outcomes

Neonatal Opioid Withdrawal Syndrome (NOWS)

Outcome ER-BUP (n=66) SL-BUP (n=69) P Value
Treated for NOWS 30.2% 26.5% .64
Opioid treatment duration 10.9 days 14.8 days .28
Hospital length of stay 8.5 days 9.5 days .54
Peak Finnegan score 10.4 10.0 .45
Head circumference at birth 34.0 cm 33.4 cm .049 ✓
12-month developmental issues 17.3% 15.4% .79

Only 28% of infants required opioid treatment for NOWS — lower than historical rates of 39–48%. All infants had live birth and were discharged alive.

Maternal Safety

Adverse Events & Safety Outcomes

Serious Adverse Events
During Pregnancy 8.7% vs 26.8%  P=.007
Post Partum 6.0% vs 18.6%  P=.04
Hospitalizations (pregnancy) 8.7% vs 26.8%
Postpartum Pain Management
Any pain medication 85.7% vs 98.5%  P=.03
Opioid pain medication 30.2% vs 50.0%  P=.02
HADS Anxiety score (PP) 5.8 vs 6.8  P=.04
Non-Serious AEs (Pregnancy)
Any non-serious TEAE 63.8% vs 66.2%
Medication-related 26.1% vs 7.0%  P=.003
GI-related (mild/moderate) Higher in ER group
Injection Site Reactions (ER only)
Severity Primarily mild–moderate
Overdose events Rare; associated with medication discontinuation
Critical Appraisal

Strengths & Limitations

Strengths
  • ✅ First RCT of ER-buprenorphine in pregnancy
  • ✅ 13 geographically diverse US sites
  • ✅ High study completion (98% through pregnancy)
  • ✅ Comprehensive effectiveness & safety data
  • ✅ Pragmatic, real-world clinical settings
  • ✅ Polysubstance use population
Limitations
  • ⚠️ Open-label design (no blinding)
  • ⚠️ Clinically stable population (most already on BUP)
  • ⚠️ Supply disruption affected 16 postpartum participants
  • ⚠️ Sample predominantly White, non-Hispanic
  • ⚠️ Some secondary outcomes underpowered
  • ⚠️ Variation in Finnegan scoring across hospitals

Funded by NIH HEAL Initiative · Extended-release buprenorphine donated by Braeburn (CAM2038/Brixadi)

Conclusions & Clinical Implications

What This Trial Tells Us

Weekly extended-release buprenorphine produced significantly higher illicit opioid abstinence during pregnancy compared to sublingual buprenorphine (82.5% vs 72.6%; P = .009), with fewer serious adverse events and less postpartum opioid pain medication use. NOWS outcomes were comparable between groups.

Winhusen TJ et al. JAMA Intern Med. Published online March 16, 2026. doi:10.1001/jamainternmed.2026.0057

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